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I-BET151 (GSK1210151A)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS842959

Background: A BET bromodomain inhibitor that interacts with BRD4 and BRD3 BET proteins and displaces them from chromatin; displays highefficacy against human and murine MLL-fusion leukemic cell lines, through the induction of early cell cycle arrest and… More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Product Name
I-BET151, Biochemical
Full Product Name
I-BET151
Product Gene Name
I-BET151 biochemical
Product Synonym Names
GSK1210151A
Form/Format
Appearance: Beige to pale yellow solid
Purity/Purification
>=98% by HPLC (>=99.5% optical purity)
Preparation and Storage
At -20 degree C
Shelf Life: 24 months
Molecular Weight
415.44
CAS Number
1300031-49-5
Structure Available?
Yes
Salt Form
No
Cell-Permeable?
Yes
MDL Number
MFCD22124472
PubChem CID
52912189
Solubility/Reconstitution Instructions
DMSO (100 mM) or Ethanol (100 mM)
SMILES
CC1=C(C(=NO1)C)C2=C(C=C3C(=C2)N=CC4=C3N(C(=O)N4)C(C)C5=CC=CC=N5)OC
InChi
InChI=1S/C23H21N5O3/c1-12-21(14(3)31-27-12)16-9-18-15(10-20(16)30-4)22-19(11-25-18)26-23(29)28(22)13(2)17-7-5-6-8-24-17/h5-11,13H,1-4H3,(H,26,29)/t13-/m1/s1
InChi Key
VUVUVNZRUGEAHB-CYBMUJFWSA-N
Handling
Protect from light and moisture

Product Categories/Family for I-BET151 biochemical

Enzyme Inhibitors; Bromodomain Inhibitors and Biochemicals; Enzyme Inhibitors; Bromodomain Inhibitors and Biochemicals (A-Z)

Structure of I-BET151 biochemical

I-BET151 GSK1210151A Biochemical – Cat# MBS842959

Other Notes

Small volumes of I-BET151 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for I-BET151 purchase

MBS842959 is a biochemical targeting I-BET151.
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