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C646, p300 / CBP Inhibitor (C646, p300/CBP Inhibitor)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS843084

Background: Cell-permeable. A reversible, p300/CBP (CREB-binding protein) histone acetyltransferase (HAT) inhibitor (Ki = 400 nM). Specific inhibition to p300 (86%) compared to N-acetyltransferase, PCAF, GCN5, Rtt109, Sas or MOZ histone acetyltransferases ( More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Product Name
C646, p300/CBP Inhibitor, Biochemical
Full Product Name
C646, p300 / CBP Inhibitor
Product Synonym Names
(E)-4-(4-((5-(4,5-Dimethyl-2-nitrophenyl)furan-2-yl)-methylene)-3-methyl-5-oxo-4,5-dihydro-1H-pyrazol-1-yl)benzoic acid
Form/Format
Appearance: Red solid
Purity/Purification
>=98% by NMR
Preparation and Storage
At -20 degree C
Shelf Life: 36 months
Molecular Weight
445.42
CAS Number
328968-36-1
Structure Available?
Yes
Salt Form
No
Cell-Permeable?
Yes
MDL Number
MFCD01784780
PubChem CID
1285941
Solubility/Reconstitution Instructions
DMSO (25 mM)
SMILES
CC1=C(C=C(C(=C1)C2=CC=C(O2)C=C3C(=NN(C3=O)C4=CC=C(C=C4)C(=O)O)C)[N+](=O)[O-])C
InChi
InChI=1S/C24H19N3O6/c1-13-10-20(21(27(31)32)11-14(13)2)22-9-8-18(33-22)12-19-15(3)25-26(23(19)28)17-6-4-16(5-7-17)24(29)30/h4-12H,1-3H3,(H,29,30)/b19-12-
InChi Key
HEKJYZZSCQBJGB-UNOMPAQXSA-N
Handling
Protect from light and air

Product Categories/Family for C646, p300/CBP Inhibitor biochemical

Biochemicals; Enzyme Inhibitors; Histone Acetyltransferase (HAT) Inhibitors and; Epigenetics; HATs; HAT Inhibitors and Biochemicals (A-Z)

Structure of C646, p300/CBP Inhibitor biochemical

C646, p300/CBP Inhibitor C646, p300 / CBP Inhibitor Biochemical – Cat# MBS843084

Other Notes

Small volumes of C646, p300/CBP Inhibitor biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for C646, p300/CBP Inhibitor purchase

MBS843084 is a biochemical targeting C646, p300/CBP Inhibitor. Also known as C646, p300 / CBP Inhibitor.
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