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GSK-690693

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS843142

Background: An ATP-competitive pan-Akt kinase inhibitor. Inhibits Akt kinase isoforms 1, 2, 3 with IC?? values of 2, 13, and 9 nM, respectively. Inhibited proliferation and induced apoptosis in a subset of tumor cells with potency consistent with… More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Product Name
GSK-690693, Biochemical
Full Product Name
GSK-690693
Product Synonym Names
4-[2-(4-Amino-1,2,5-oxadiazol-3-yl)--1-ethyl-7-[(3S)-3-piperidinylmethoxy)-1H-imidazo[-4,5-c]pyridin-4-yl]-2-methyl-3-butyn-2-ol
Form/Format
Appearance: Yellow solid
Purity/Purification
>=98% by HPLC
Preparation and Storage
At -20 degree C
Shelf Life: 24 months
Molecular Weight
425.48
CAS Number
937174-76-0
Structure Available?
Yes
Salt Form
No
Cell-Permeable?
Yes
MDL Number
MFCD14105605
PubChem CID
16725726
Solubility/Reconstitution Instructions
DMSO (~20 mg/ml)
SMILES
CCN1C2=C(C(=NC=C2OCC3CCCNC3)C#CC(C)(C)O)N=C1C4=NON=C4N
InChi
InChI=1S/C21H27N7O3/c1-4-28-18-15(30-12-13-6-5-9-23-10-13)11-24-14(7-8-21(2,3)29)16(18)25-20(28)17-19(22)27-31-26-17/h11,13,23,29H,4-6,9-10,12H2,1-3H3,(H2,22,27)/t13-/m0/s1
InChi Key
KGPGFQWBCSZGEL-ZDUSSCGKSA-N
Handling
Protect from air and moisture

Product Categories/Family for GSK-690693 biochemical

Enzyme Inhibitors; Protein Kinase Inhibitors; Akt Inhibitors and Biochemicals; Enzyme Inhibitors; Protein Kinase Inhibitors and Biochemicals (A-Z)

Structure of GSK-690693 biochemical

GSK-690693 Biochemical – Cat# MBS843142

Other Notes

Small volumes of GSK-690693 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for GSK-690693 purchase

MBS843142 is a biochemical targeting GSK-690693.
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