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ARN-509

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS845717

ARN-509 is a selective and competitive androgen receptor (AR) inhibitor (IC50 = 16 nM). ARN-509 selectively binds the androgen receptor and impairs its nuclear translocation and DNA binding to androgen response elements useful for prostate cancer treatment. More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Product Name
ARN-509, Biochemical
Full Product Name
ARN-509
Product Gene Name
ARN-509 biochemical
Product Synonym Names
4-[7-[6-cyano-5- (trifluoromethyl) pyridin-3-yl]-8-oxo-6-sulfanylidene-5; 7-diazaspiro[3.4]octan-5-yl]-2-fluoro-N-methylbenzamide
Form/Format
White to off-white solid
Purity/Purification
>=98% by HPLC
Preparation and Storage
Store at -20 degree C for 36 months.
Protect from air and light.
Molecular Weight
477.43
Salt Form
No
Molecular Formula
C21H15F4N5O2S
CAS Number
956104-40-8
Cell-Permeable
Yes
Reconstitution
DMSO (>5 mg/ml)
SMILES
NC(=O)C1=C(C=C(C=C1)N2C(=S)N(C(=O)C23CCC3)C4=CN=C(C(=C4)C(F)(F)F)C#N)F
InChi
InChI=1S/C21H15F4N5O2S/c1-27-17(31)13-4-3-11(8-15(13)22)30-19(33)29(18(32)20(30)5-2-6-20)12-7-14(21(23,24)25)16(9-26)28-10-12/h3-4,7-8,10H,2,5-6H2,1H3,(H,27,31)
InChi Key
HJBWBFZLDZWPHF-UHFFFAOYSA-N

Structure of ARN-509 biochemical

ARN-509 Biochemical – Cat# MBS845717

Other Notes

Small volumes of ARN-509 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for ARN-509 purchase

MBS845717 is a biochemical targeting ARN-509.
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