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EPZ015866 (GSK591)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS846358

EPZ015866 (GSK591) is a potent selective inhibitor of the arginine methyltransferase PRMT5/MEP50 complex thus stopping the methylation of histone H4 with IC50 of 11 nM. It also maintains superior selectivity against other panels of methyl transferases… More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Product Name
EPZ015866, Biochemical
Full Product Name
EPZ015866 (GSK591)
Product Gene Name
EPZ015866 biochemical
Product Synonym Names
(S)-2- (cyclobutylamino)-N- (3- (3; 4-dihydroisoquinolin-2 (1H)-yl)-2-hydroxypropyl) isonicotinamide
Form/Format
Crystalline solid
Purity/Purification
>=98% by HPLC
Preparation and Storage
Store at -20 degree C for 36 months.
Protect from air and light.
Molecular Weight
380.5
Salt Form
No
Molecular Formula
C22H28N4O2
CAS Number
1616391-87-7
Cell-Permeable
Yes
Reconstitution
DMSO (>40 mg/ml)
SMILES
C1CC(C1)NC2=NC=CC(=C2)C(=O)NCC(CN3CCC4=CC=CC=C4C3)O
InChi
InChI=1S/C22H28N4O2/c27-20(15-26-11-9-16-4-1-2-5-18(16)14-26)13-24-22(28)17-8-10-23-21(12-17)25-19-6-3-7-19/h1-2,4-5,8,10,12,19-20,27H,3,6-7,9,11,13-15H2,(H,23,25)(H,24,28)/t20-/m0/s1
InChi Key
TWKYXZSXXXKKJU-FQEVSTJZSA-N

Structure of EPZ015866 biochemical

EPZ015866 (GSK591) Biochemical – Cat# MBS846358

Other Notes

Small volumes of EPZ015866 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for EPZ015866 purchase

MBS846358 is a biochemical targeting EPZ015866. Also known as EPZ015866 (GSK591).
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