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BX-912

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS848098

BX-912 is a potent and selective inhibitor of 3-phosphoinositide-dependent kinase 1 (PDK1) with IC50 value of 26nM. BX-912 has shown 9-fold selectivity for PDK1 relative to PKA and 105-fold selectivity against PKC. More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Product Name
BX-912, Biochemical
Full Product Name
BX-912
Product Synonym Names
BX-912; BX 912; BX912; N-[3-[[5-bromo-4-[2- (1H-imidazol-5-yl) ethylamino]pyrimidin-2-yl]amino]phenyl]pyrrolidine-1-carboxamide; N- (3- ( (4- ( (2- (1H-imidazol-4-yl) ethyl) amino)-5-bromopyrimidin-2-yl) amino) phenyl) pyrrolidine-1-carboxamide; PDK1 inhibitor
Form/Format
Solid powder
Purity/Purification
>98%
Preparation and Storage
Store at -20 degree C
Protect from air and light
Shelf life: ~36 months
Molecular Weight
471.35
Solubility
DMSO
Molecular Formula
C??H??BrN?O
CAS Number
702674-56-4
MDL Number
MFCD10565925
PubChem CID
11754511
SMILES
C1CCN (C1)C (=O)NC2=CC=CC (=C2)NC3=NC=C (C (=N3)NCCC4=CN=CN4)Br
InChi
InChI=1S/C20H23BrN8O/c21-17-12-24-19 (28-18 (17)23-7-6-16-11-22-13-25-16)26-14-4-3-5-15 (10-14)27-20 (30)29-8-1-2-9-29/h3-5,10-13H,1-2,6-9H2, (H,22,25)(H,27,30)(H2,23,24,26,28)
InChi Key
DMMILYKXNCVKOJ-UHFFFAOYSA-N

Product Categories/Family for BX-912 biochemical

Enzyme Inhibitors; Protein Kinase Inhibitors; mTOR Inhibitors; Enzyme Inhibitors (A-Z); Signaling Pathways; PI3 K; Akt; mTOR Signaling; Inhibitors; Biochemicals; Biochemicals (A-Z)

Structure of BX-912 biochemical

Bx-912 Biochemical – Cat# MBS848098

Product References and Citations for BX-912 biochemical

https://pubchem.ncbi.nlm.nih.gov/compound/11754511

Other Notes

Small volumes of BX-912 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for BX-912 purchase

MBS848098 is a biochemical targeting BX-912.
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