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MSC-2530818

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS848270

MSC-2530818 is a potent, selective CDK8 Inhibitor (IC50 = 2.6 nM). It displays potent inhibition of phospho-STAT1SER727, an established biomarker of CDK8 activity. MSC2530818 demonstrates potent inhibition of WNT-dependent transcription in human cancer cell… More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Product Name
MSC-2530818, Biochemical
Full Product Name
MSC-2530818
Product Synonym Names
[ (2S)-2- (4-Chlorophenyl) pyrrolidin-1-yl]- (3-methyl-1H-pyrazolo[3; 4-b]pyridin-5-yl) methanone
Form/Format
Crystalline solid
Purity/Purification
>=98% by HPLC
Preparation and Storage
Store at -20 degree C
Protect from air and light
Shelf life: ~36 months
Molecular Weight
340.81
Solubility
DMSO (~ 5 mg/ml)
Molecular Formula
C??H??ClN?O 
CAS Number
1883423-59-3 
PubChem CID
118879529
SMILES
CC1=C2C=C (C=NC2=NN1)C (=O)N3CCCC3C4=CC=C (C=C4)Cl
InChi
InChI=1S/C18H17ClN4O/c1-11-15-9-13 (10-20-17 (15)22-21-11)18 (24)23-8-2-3-16 (23)12-4-6-14 (19)7-5-12/h4-7,9-10,16H,2-3,8H2,1H3, (H,20,21,22)/t16-/m0/s1
InChi Key
ODRITQGYYWHQGM-INIZCTEOSA-N

Product Categories/Family for MSC-2530818 biochemical

Enzyme Inhibitors; Protein Kinase Inhibitors; CDK Inhibitors; Enzyme Inhibitors (A-Z); Biochemicals; Biochemicals (A-Z)

Structure of MSC-2530818 biochemical

MSC-2530818 Biochemical – Cat# MBS848270

Product References and Citations for MSC-2530818 biochemical

https://pubchem.ncbi.nlm.nih.gov/compound/118879529

Other Notes

Small volumes of MSC-2530818 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for MSC-2530818 purchase

MBS848270 is a biochemical targeting MSC-2530818.
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