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ARV-825

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS848312

ARV-825 is a BRD4 inhibitor. It is a hetero-bifunctional PROTAC (Proteolysis Targeting Chimera) that recruits BRD4 to the E3 ubiquitin ligase cereblon, leading to fast, efficient, and prolonged degradation of BRD4. ARV-825 more effectively suppresses c-MYC… More details

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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Product Overview

Product Name
ARV-825, Biochemical
Full Product Name
ARV-825
Product Synonym Names
2- ( (S)-4- (4-chlorophenyl)-2; 3; 9-trimethyl-6H-thieno[3; 2-f][1; 2; 4]triazolo[4; 3-a][1; 4]diazepin-6-yl)-N- (4- (2- (2- (2- (2- ( (2- (2; 6-dioxopiperidin-3-yl)-1; 3-dioxoisoindolin-4-yl) amino) ethoxy) ethoxy) ethoxy) ethoxy) phenyl) acetamide
Form/Format
Crystalline solid
Purity/Purification
>98% by HPLC
Preparation and Storage
Store at -20 degree C
Protect from air and light
Shelf life: ~36 months
Molecular Weight
941.4
Solubility
DMSO
Molecular Formula
C??H??ClN?O?S
CAS Number
1818885-28-7
PubChem CID
92044400
SMILES
CC1=C (SC2=C1C (=NC (C3=NN=C (N32)C)CC (=O)NC4=CC=C (C=C4)OCCOCCOCCOCCNC5=CC=CC6=C5C (=O)N (C6=O)C7CCC (=O)NC7=O)C8=CC=C (C=C8)Cl)C
InChi
InChI=1S/C46H47ClN8O9S/c1-26-27 (2)65-46-39 (26)41 (29-7-9-30 (47)10-8-29)50-35 (42-53-52-28 (3)54 (42)46)25-38 (57)49-31-11-13-32 (14-12-31)64-24-23-63-22-21-62-20-19-61-18-17-48-34-6-4-5-33-40 (34)45 (60)55 (44 (33)59)36-15-16-37 (56)51-43 (36)58/h4-14,35-36,48H,15-25H2,1-3H3, (H,49,57)(H,51,56,58)/t35-,36/m0/s1
InChi Key
RWLOGRLTDKDANT-TYIYNAFKSA-N

Product Categories/Family for ARV-825 biochemical

Epigenetics; Epigenetic Modulators (A-Z); Biochemicals; Biochemicals (A-Z)

Structure of ARV-825 biochemical

ARV-825 Biochemical – Cat# MBS848312

Product References and Citations for ARV-825 biochemical

https://pubchem.ncbi.nlm.nih.gov/compound/92044400

Other Notes

Small volumes of ARV-825 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for ARV-825 purchase

MBS848312 is a biochemical targeting ARV-825.
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