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AZD-5153

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS848313

AZD-5153 is a potent, selective, and orally available BET/BRD4 bromodomain inhibitor with a bivalent binding mode. AZD-5153 ligates two bromodomains in BRD4 simultaneously. Displays cellular and antitumor activity in preclinical hematologic tumor models. More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Product Name
AZD-5153, Biochemical
Full Product Name
AZD-5153
Product Synonym Names
4-[2-[4-[1- (3-methoxy-[1; 2; 4]triazolo[4; 3-b]pyridazin-6-yl) piperidin-4-yl]phenoxy]ethyl]-1; 3-dimethylpiperazin-2-one; 6-hydroxynaphthalene-2-carboxylic acid
Form/Format
Crystalline solid
Purity/Purification
>=98% by HPLC
Preparation and Storage
Store at -20 degree C
Protect from air and light
Shelf life: ~36 months
Molecular Weight
667.8
Solubility
DMSO
Molecular Formula
C??H??N?O? ?C??H?O?
CAS Number
1869912-40-2
PubChem CID
126970641
SMILES
CC1C (=O)N (CCN1CCOC2=CC=C (C=C2)C3CCN (CC3)C4=NN5C (=NN=C5OC)C=C4)C.C1=CC2=C (C=CC (=C2)O)C=C1C (=O)O
InChi
InChI=1S/C25H33N7O3.C11H8O3/c1-18-24 (33)29 (2)14-15-30 (18)16-17-35-21-6-4-19 (5-7-21)20-10-12-31 (13-11-20)23-9-8-22-26-27-25 (34-3)32 (22)28-23;12-10-4-3-7-5-9 (11 (13)14)2-1-8 (7)6-10/h4-9,18,20H,10-17H2,1-3H3;1-6,12H, (H,13,14)
InChi Key
UNZQBHXKCHECEC-UHFFFAOYSA-N

Product Categories/Family for AZD-5153 biochemical

Epigenetics; Epigenetic Modulators (A-Z); Biochemicals; Biochemicals (A-Z)

Structure of AZD-5153 biochemical

AZD-5153 Biochemical – Cat# MBS848313

Product References and Citations for AZD-5153 biochemical

https://pubchem.ncbi.nlm.nih.gov/compound/126970641#section=Top

Other Notes

Small volumes of AZD-5153 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for AZD-5153 purchase

MBS848313 is a biochemical targeting AZD-5153.
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