ACT-129968 (Setipiprant)

Name: ACT-129968 (Setipiprant); MyBioSource
Brand: MyBioSource
SKU: MBS848593
Price: 210 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS848593

A potent and selective CRTh2 antagonist. CRTh2 is a G-protein-coupled receptor for prostaglandin D2 (PGD2), a key mediator in inflammatory disorders. More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Product Name

ACT-129968, Biochemical

Full Product Name

ACT-129968

Product Synonym Names

Setipiprant; 2- (2- (1-naphthoyl)-8-fluoro-1; 2; 3; 4-tetrahydro-5H-pyrido[4; 3-b]indol-5-yl) acetic acid

Form/Format

Crystalline solid

Purity/Purification

>=98% by HPLC

Preparation and Storage

Store at -20 degree C
Shelf life: ~36 months

Molecular Weight

402.43

Solubility

>30 mg/ml

Molecular Formula

C??H??FN?O?

CAS Number

866460-33-5

PubChem CID

49843471

SMILES

C1CN (CC2=C1N (C3=C2C=C (C=C3)F)CC (=O)O)C (=O)C4=CC=CC5=CC=CC=C54

InChi

InChI=1S/C24H19FN2O3/c25-16-8-9-21-19 (12-16)20-13-26 (11-10-22 (20)27 (21)14-23 (28)29)24 (30)18-7-3-5-15-4-1-2-6-17 (15)18/h1-9,12H,10-11,13-14H2, (H,28,29)

InChi Key

IHAXLPDVOWLUOS-UHFFFAOYSA-N

Product Categories/Family for ACT-129968 biochemical

Biochemicals; Enzyme Inhibitors; Other Inhibitors; Enzyme Inhibitors (A-Z); Biochemicals (A-Z)

Product References and Citations for ACT-129968 biochemical

https://pubchem.ncbi.nlm.nih.gov/compound/49843471

Other Notes

Small volumes of ACT-129968 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for ACT-129968 purchase

MBS848593 is a biochemical targeting ACT-129968.