Etrasimod (APD-334)

Name: Etrasimod (APD-334); MyBioSource
Brand: MyBioSource
SKU: MBS848596
Price: 265 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS848596

A potent and selective sphingosine-1-phosphate-1 (S1P1) receptor antagonist (IC50 =1.88 nM in CHO cells) . More details

DISCONTINUED
Click here to view our similar product(s) OR click here to contact our technical support team for suitable replacement.

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Product Name

Etrasimod, Biochemical

Full Product Name

Etrasimod

Product Synonym Names

APD-334; (3R)-7-[[4-cyclopentyl-3- (trifluoromethyl) phenyl]methoxy]-1; 2; 3; 4-tetrahydro-cyclopent[b]indole-3-acetic acid; APD334

Form/Format

Crystalline solid

Purity/Purification

>=98%

Preparation and Storage

Store at -20 degree C
Shelf life: ~12 months

Molecular Weight

457.49

Solubility

>25 mg/ml (DMSO)

Molecular Formula

C??H??F?NO?

CAS Number

1206123-37-6

PubChem CID

44623998

SMILES

C1CCC (C1)C2=C (C=C (C=C2)COC3=CC4=C (C=C3)NC5=C4CCC5CC (=O)O)C (F)(F)F

InChi

InChI=1S/C26H26F3NO3/c27-26 (28,29)22-11-15 (5-8-19 (22)16-3-1-2-4-16)14-33-18-7-10-23-21 (13-18)20-9-6-17 (12-24 (31)32)25 (20)30-23/h5,7-8,10-11,13,16-17,30H,1-4,6,9,12,14H2, (H,31,32)/t17-/m1/s1

InChi Key

MVGWUTBTXDYMND-QGZVFWFLSA-N

Product Categories/Family for Etrasimod biochemical

Enzyme Inhibitors; Protein Kinase Inhibitors; Protein Kinase Inhibitors (A-Z); Biochemicals (A-Z); Other Inhibitors; Enzyme Inhibitors (A-Z)

Product References and Citations for Etrasimod biochemical

https://pubchem.ncbi.nlm.nih.gov/compound/44623998

Other Notes

Small volumes of Etrasimod biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Etrasimod purchase

MBS848596 is a biochemical targeting Etrasimod.