GSK-5959 (N-[2)

Name: GSK-5959 (N-[2); MyBioSource
Brand: MyBioSource
SKU: MBS848619
Price: 210 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS848619

GSK-5959 is a potent and selective BRPF1 (BR140 or Peregrin) bromodomain inhibitor (IC50 = 80 nM). GSK-5959 displays >100-fold selectivity for BRPF1 over a panel of 35 other bromodomains. BRPF1 (bromodomain and PHD finger containing protein 1) is involved in… More details

DISCONTINUED
Click here to view our similar product(s) OR click here to contact our technical support team for suitable replacement.

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Product Name

GSK-5959, Biochemical

Full Product Name

GSK-5959

Product Synonym Names

N-[2; 3-Dihydro-1; 3-dimethyl-2-oxo-6- (1-piperidinyl)-1H-benzimidazol-5-yl]-2-methoxybenzamide; GSK5959

Form/Format

Pale yellow solid

Purity/Purification

>=98% by HPLC

Preparation and Storage

Store at -20 degree C
Shelf life: ~36 months

Molecular Weight

394.47

Solubility

~4 mg/ml (DMSO)

Molecular Formula

C??H??N?O?

CAS Number

901245-65-6

PubChem CID

15990224

SMILES

CN1C2=CC (=C (C=C2N (C1=O)C)N3CCCCC3)NC (=O)C4=CC=CC=C4OC

InChi

InChI=1S/C22H26N4O3/c1-24-18-13-16 (23-21 (27)15-9-5-6-10-20 (15)29-3)17 (26-11-7-4-8-12-26)14-19 (18)25 (2)22 (24)28/h5-6,9-10,13-14H,4,7-8,11-12H2,1-3H3, (H,23,27)

InChi Key

LTUGYAOMCKNTGG-UHFFFAOYSA-N

Product Categories/Family for GSK-5959 biochemical

Enzyme Inhibitors; Enzyme Inhibitors (A-Z); Biochemicals; Biochemicals (A-Z); Cancer Research; Epigenetic Regulation; Reader Domains; Bromodomains; Bromodomain Inhibitors; Epigenetic Modulators (A-Z)

Product References and Citations for GSK-5959 biochemical

https://pubchem.ncbi.nlm.nih.gov/compound/15990224

Other Notes

Small volumes of GSK-5959 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for GSK-5959 purchase

MBS848619 is a biochemical targeting GSK-5959.