SSR-240612 ((3R)-3- (1)

Name: SSR-240612 ((3R)-3- (1); MyBioSource
Brand: MyBioSource
SKU: MBS848625
Price: 210 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS848625

SSR-240612 is a potent and selective, non-peptide antagonist of the bradykinin B1 receptor (Kis = 0.48-0.73 and 358-481 nM for B1 and B2 receptors, respectively). It inhibits the contraction of rabbit aorta and rat ileum induced by the B1 receptor agonist… More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Product Name

SSR-240612, Biochemical

Full Product Name

SSR-240612

Product Synonym Names

(3R)-3- (1; 3-benzodioxol-5-yl)-N-[ (6-methoxy-2-naphthalenyl) sulfonyl]-beta-alanyl-4-[[ (2R; 6S)-2; 6-dimethyl-1-piperidinyl]methyl]-N-methyl-N- (1-methylethyl)-D-phenylalaninamide; monohydrochloride

Form/Format

Crystalline solid

Purity/Purification

>=98% by HPLC

Preparation and Storage

Store at -20 degree C
Shelf life: ~36 months

Molecular Weight

793.4

Solubility

>25 mg/ml (DMSO)

Molecular Formula

C??H??N?O?S- HCl

CAS Number

464930-42-5

PubChem CID

44235958

SMILES

CC1CCCC (N1CC2=CC=C (C=C2)CC (C (=O)N (C)C (C)C)NC (=O)CC (C3=CC4=C (C=C3)OCO4)NS (=O)(=O)C5=CC6=C (C=C5)C=C (C=C6)OC)C.Cl

InChi

InChI=1S/C42H52N4O7S.ClH/c1-27 (2)45 (5)42 (48)38 (20-30-10-12-31 (13-11-30)25-46-28 (3)8-7-9-29 (46)4)43-41 (47)24-37 (34-16-19-39-40 (23-34)53-26-52-39)44-54 (49,50)36-18-15-32-21-35 (51-6)17-14-33 (32)22-36;/h10-19,21-23,27-29,37-38,44H,7-9,20,24-26H2,1-6H3, (H,43,47);1H/t28-,29+,37-,38-;/m1./s1

InChi Key

GLHHFOSVBQQNAW-GDYXXZBVSA-N

Product Categories/Family for SSR-240612 biochemical

Biochemicals; Enzyme Inhibitors; Other Inhibitors; Enzyme Inhibitors (A-Z); Biochemicals (A-Z)

Product References and Citations for SSR-240612 biochemical

https://pubchem.ncbi.nlm.nih.gov/compound/44235958#section=Top

Other Notes

Small volumes of SSR-240612 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for SSR-240612 purchase

MBS848625 is a biochemical targeting SSR-240612.