LP99 (N-[ (2R)

Name: LP99 (N-[ (2R); MyBioSource
Brand: MyBioSource
SKU: MBS848988
Price: 205 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS848988

LP99 is an inhibitor of BRD9 and BRD7 bromodomains. LP99 inhibits the interactions of both BRD7 and BRD9 with histones H3.3 and H4, with IC50 values in the low micromolar range in bioluminescence resonance energy transfer (BRET) assays in HEK293 cells. It… More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Product Name

LP99, Biochemical

Full Product Name

LP99

Product Synonym Names

N-[ (2R; 3S)-2- (4-chlorophenyl)-1- (1; 4-dimethyl-2-oxoquinolin-7-yl)-6-oxopiperidin-3-yl]-2-methylpropane-1-sulfonamide; N-[ (2R; 3S)-2- (4-chlorophenyl)-1- (1; 2-dihydro-1; 4-dimethyl-2-oxo-7-quinolinyl)-6-oxo-3-piperidinyl]-2-methyl-1-propanesulfonamide

Form/Format

A crystalline solid

Purity/Purification

>=98%

Preparation and Storage

Store at -20 degree C
Shelf life: ~36 months

Molecular Weight

516.05

Solubility

~20 mg/ml in ethanol
DMSO and DMF

Molecular Formula

C??H??ClN?O?S

CAS Number

1808951-93-0

PubChem CID

91827372

SMILES

CC1=CC (=O)N (C2=C1C=CC (=C2)N3C (C (CCC3=O)NS (=O)(=O)CC (C)C)C4=CC=C (C=C4)Cl)C

InChi

InChI=1S/C26H30ClN3O4S/c1-16 (2)15-35 (33,34)28-22-11-12-24 (31)30 (26 (22)18-5-7-19 (27)8-6-18)20-9-10-21-17 (3)13-25 (32)29 (4)23 (21)14-20/h5-10,13-14,16,22,26,28H,11-12,15H2,1-4H3/t22-,26+/m0/s1

InChi Key

LVDRREOUMKACNJ-BKMJKUGQSA-N

Product Categories/Family for LP99 biochemical

Biochemicals; Biochemicals (A-Z); Cancer Research; Epigenetic Regulation; Reader Domains; Bromodomains; Bromodomain Inhibitors; Biochemicals; Enzyme Inhibitors; Enzyme Inhibitors (A-Z)

Product References and Citations for LP99 biochemical

https://pubchem.ncbi.nlm.nih.gov/compound/91827372

Other Notes

Small volumes of LP99 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for LP99 purchase

MBS848988 is a biochemical targeting LP99.