GLPG-1690 (Ziritaxestat)

Name: GLPG-1690 (Ziritaxestat); MyBioSource
Brand: MyBioSource
SKU: MBS3602426
Price: 235 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3602426

GLPG-1690 (Ziritaxestat, GLPG1690) is a first-in-class, potent, competitive autotaxin inhibitor with Ki/IC50 of 15 nM/131 nM. More details

$235 / 5 mg +1 FREE 8GB USB

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

GLPG-1690, Biochemical

Full Product Name

GLPG-1690

Product Synonym Names

Ziritaxestat; GLPG 1690; GLPG1690

Purity/Purification

>98% (HPLC)

Preparation and Storage

Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack

Molecular Weight

588.71

Suitability

DMSO: Soluble (<1mg/mL refers to the product slightly soluble or insoluble)

Target

Autotaxin

Receptor

autotaxin

Chemical Name

2-[[2-Ethyl-6-[4-[2-(3-hydroxyazetidin-1-yl)-2-oxoethyl]-piperazin-1-yl]-8-methylimidazo[1, 2-a]pyridin-3-yl]-methylamino]-4-(4-fluorophenyl)thiazole-5-carbonitrile

SMILES

CCC(N=C1N2C=C(C=C1C)N3CCN(CC3)CC(N4CC(C4)O)=O)=C2N(C)C5=NC(C6=CC=C(C=C6)F)=C(S5)C#N

Molecular Formula

C30H33FN8O2S

CAS Number

1628260-79-6

Product Categories/Family for GLPG-1690 biochemical

Fibrosis; Wnt/Notch/Hedgehog; Other Indications

Product References and Citations for GLPG-1690 biochemical

1. Desroy N, et al. J Med Chem. 2017 May 11; 60 (9):3580-3590.

Other Notes

Small volumes of GLPG-1690 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for GLPG-1690 purchase

MBS3602426 is a biochemical targeting GLPG-1690.