• Call +1.858.633.0165 or Fax +1.858.633.0166 or Contact Us

GAT-100

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3602537

GAT-100 (GAT100) is a potent, selective CB1R negative allosteric modulator (NAM) with cAMP EC50 and beta-arr EC50 of 174 nM and 2.1 nM. More details

$1025 / 5 mg +1 FREE 8GB USB
Product Documentation
PDF
Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
GAT-100, Biochemical
Full Product Name
GAT-100
Product Synonym Names
GAT100
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
432.59
Target
Cannabinoid Receptor
Receptor
Cannabinoid Receptor
Chemical Name
3-Ethyl-5-isothiocyanato-N-(4-(piperidin-1-yl)phenethyl)-1H-indole-2-carboxamide
SMILES
O=C(C(N1)=C(CC)C2=C1C=CC(N=C=S)=C2)NCCC3=CC=C(N4CCCCC4)C=C3
Molecular Formula
C25H28N4OS
CAS Number
1663564-42-8

Product Categories/Family for GAT-100 biochemical

GPCR/G Protein

Structure of GAT-100 biochemical

GAT-100 Biochemical – Cat# MBS3602537

Product References and Citations for GAT-100 biochemical

1. Kulkarni PM, et al. J Med Chem. 2016 Jan 14; 59 (1):44-60.
2. Laprairie RB, et al. ACS Chem Neurosci. 2016 Jun 15; 7 (6):776-98.

Other Notes

Small volumes of GAT-100 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for GAT-100 purchase

MBS3602537 is a biochemical targeting GAT-100.
Request a Quote

Please fill out the form below and our representative will get back to you shortly.

MBS000000
Contact Us

Please fill out the form below and our representative will get back to you shortly.

MBS000000