Anacetrapib (MK 0859)

Name: Anacetrapib (MK 0859); MyBioSource
Brand: MyBioSource
SKU: MBS3606357
Price: 215 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3606357

Anacetrapib (MK 0859) is a potent, orally active cholesteryl ester transfer protein (CETP) inhibitor with IC50 of 7.9 nM and 11.8 nM for rhCETP and C13S CETP mutant, respectively. More details

$215 / 2 mg +1 FREE 8GB USB

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Anacetrapib, Biochemical

Full Product Name

Anacetrapib

Product Synonym Names

MK 0859; MK-0859; MK0859

Purity/Purification

>98% (HPLC)

Preparation and Storage

Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack

Molecular Weight

637.5084

Suitability

10mM in DMSO

Target

CETP

Receptor

MutantCETP (C13S); rhCETP

Chemical Name

2-Oxazolidinone, 5-[3, 5-bis(trifluoromethyl)phenyl]-3-[[4'-fluoro-2'-methoxy-5'-(1-methylethyl)-4-(trifluoromethyl)[1, 1'-biphenyl]-2-yl]methyl]-4-methyl-, (4S, 5R)

SMILES

O=C1O[C@H](C2=CC(C(F)(F)F)=CC(C(F)(F)F)=C2)[C@H](C)N1CC3=CC(C(F)(F)F)=CC=C3C4=CC(C(C)C)=C(F)C=C4OC

Molecular Formula

C30H25F10NO3

CAS Number

875446-37-0

Product Categories/Family for Anacetrapib biochemical

Atherosclerosis; Metabolic Enzyme/Protease; Cardiovascular Disease

Product References and Citations for Anacetrapib biochemical

1. Krishna R, et al. Lancet. 2007 Dec 8; 370 (9603):1907-14.
2. Vergeer M, et al. Nat Clin Pract Cardiovasc Med. 2008 Jun; 5 (6):302-3.
3. Cannon CP, et al. Am Heart J. 2009 Oct; 158 (4):513-519.e3.
4. Niesor EJ, et al. J Lipid Res. 2010 Dec; 51 (12):3443-54.

Other Notes

Small volumes of Anacetrapib biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Anacetrapib purchase

MBS3606357 is a biochemical targeting Anacetrapib.