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ERK5-IN-1

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3609943

ERK5-IN-1 is a potent ERK5 inhibitor (IC50: 87 nM). It also inhibits LRRK2[G2019S] (IC50: 26 nM). More details

$290 / 5 mg +1 FREE 8GB USB
Product Documentation
PDF
Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
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Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
ERK5-IN-1, Biochemical
Full Product Name
ERK5-IN-1
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
459.54
Suitability
DMSO: 10mM
Target
ERK
Receptor
ERK5
Chemical Name
6H-Pyrimido[45-b][14]benzodiazepin-6-one 511-dihydro-2-[[2-methoxy-4-(4-methyl-1-piperazinyl)phenyl]amino]-511-dimethyl
SMILES
COc1cc(ccc1Nc1ncc2N(C)C(=O)c3ccccc3N(C)c2n1)N1CCN(C)CC1
Molecular Formula
C25H29N7O2
CAS Number
1234479-76-5

Product Categories/Family for ERK5-IN-1 biochemical

MAPK/ERK Signaling

Structure of ERK5-IN-1 biochemical

ERK5-IN-1 Biochemical – Cat# MBS3609943

Product References and Citations for ERK5-IN-1 biochemical

1.Deng X et al. Structural determinants for ERK5 (MAPK7) and leucine rich repeat kinase 2 activities of benzo [e]pyrimido- [54-b]diazepine-6 (11H)-ones. Eur J Med Chem. 2013; 70:758-767.

Other Notes

Small volumes of ERK5-IN-1 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for ERK5-IN-1 purchase

MBS3609943 is a biochemical targeting ERK5-IN-1.
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