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GSK2193874

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3610309

MBS3610309 is a biochemical targeting GSK2193874. GSK2193874 was identified as a selective orally active TRPV4 blocker. More details

$235 / 2 mg +1 FREE 8GB USB
Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
GSK2193874, Biochemical
Full Product Name
GSK2193874
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
691.6
Suitability
DMSO: 100mg/mL (144.59mM)
Target
TRP/TRPV Channel
Receptor
TRPV4
Chemical Name
7-bromo-N-(1-phenylcyclopropyl)-3-[(4-piperidin-1-ylpiperidin-1-yl) methyl]-2-[3-(trifluoromethyl)phenyl]quinoline-4-carboxamide
SMILES
FC(F)(F)c1cccc(c1)-c1nc2cc(Br)ccc2c(C(=O)NC2(CC2)c2ccccc2)c1CN1CCC(CC1)N1CCCCC1
Molecular Formula
C37H38BrF3N4O
CAS Number
1336960-13-4

Product Categories/Family for GSK2193874 biochemical

Membrane Transporter/Ion Channel

Product References and Citations for GSK2193874 biochemical

1.Cheung M Bao W Behm D J et al. Discovery of GSK2193874: An Orally Active Potent and Selective Blocker of Transient Receptor Potential Vanilloid 4 [J]. ACS Medicinal Chemistry Letters 2017:acsmedchemlett.7b00094.

Other Notes

Small volumes of GSK2193874 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.
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