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ARN272 Inhibitor – ARN 272

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5751779

MBS5751779 is an inhibitor targeting ARN272. Also known as ARN 272. ARN272 is a FAAH-like anandamide transporter (FLAT) inhibitor (IC50: 1.8uM). More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
ARN 272 (ARN272), Inhibitor
Full Product Name
ARN 272
Product Gene Name
ARN272, inhibitor
Form/Format
Powder
Purity/Purification
98.23%
Preparation and Storage
Store at -20 degree C for 3 years powder; -80 degree C for 2 years in solvent
For obtaining a higher solubility, please warm the tube at 37 degree C and shake it in the ultrasonic bath for a while. Stock solution can be stored below -20 degree C for several month.
Molecular Weight
432.47
Formula
C27H20N4O2
CAS
488793-85-7
Smiles
Oc1ccc(cc1)-c1nnc(Nc2ccc(cc2)C(=O)Nc2ccccc2)c2ccccc12
Receptor (IC50)
anandamide transporter: 1.8uM
Solubility
DMSO: 50mg/mL, 115.61mM
Ethanol: 8mg/mL, 18.50mM
Water: Insoluble
(<1mg/ml refers to the product slightly soluble or insoluble)

Product Categories/Family for ARN272, inhibitor

Home; Others

Structure of ARN272, inhibitor

ARN272 Inhibitor – Cat# MBS5751779

Product References and Citations for ARN272, inhibitor

1. Fu J, et al. A catalytically silent FAAH-1 variant drives anandamide transport in neurons. Nat Neurosci. 2011 Nov 20;15 (1):64-9.
2. O'Brien LD, et al. Anandamide transport inhibition by ARN272 attenuates nausea-induced behaviour in rats, and vomiting in shrews (Suncus murinus). Br J Pharmacol. 2013 Nov;170 (5):1130-6.

Other Notes

Small volumes of ARN272, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.
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