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GCN2-IN-1 Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5753170

GCN2-IN-1 (A-92) is a potent general control nonderepressible 2 kinase (GCN2) inhibitor with an IC50 of 0.3-3uM in the cell assay and an IC50 of More details

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Product Documentation
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Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
GCN2-IN-1, Inhibitor
Full Product Name
GCN2-IN-1
Product Gene Name
GCN2-IN-1, inhibitor
Product Synonym Names
A-92
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
402.41
Solubility
DMSO: 60mg/mL (149.10mM) Need ultrasonic and warming
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C19H18N10O
SMILES
C1(NC2=CN(C3CCOCC3)N=C2)=NC=C(N=NN4C5=CC6=C(C=C5)C=NN6)C4=N1
CAS Number
1448693-69-3
Target & IC50
GCN2: ic50 <0.3uM

Structure of GCN2-IN-1, inhibitor

GCN2-IN-1 Inhibitor – Cat# MBS5753170

Product References and Citations for GCN2-IN-1, inhibitor

Dieter Dorsch, et al. Triazolo[4,5-d]pyrimidine derivatives. WO2013110309A1.
Dieter Dorsch, et al. Triazolo[4,5-d]pyrimidine derivatives. WO2013110309A1.

Other Notes

Small volumes of GCN2-IN-1, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for GCN2-IN-1 purchase

MBS5753170 is an inhibitor targeting GCN2-IN-1.
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