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PSB-12379 Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5753736

PSB-12379 is a potent inhibitor of Ecto-5'-Nucleotidase (CD73)(Kis of 9.03nM (rat) and 2.21nM (human)). More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Product Name
PSB-12379, Inhibitor
Full Product Name
PSB-12379
Product Gene Name
PSB-12379, inhibitor
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
515.35
Solubility
H2O: 7.14mg/mL (13.85mM) Need ultrasonic
DMSO: <1mg/mL (insoluble or slightly soluble)
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C18H23N5O9P2
SMILES
O[C@@H]([C@H]1O)[C@@H](COP(CP(O)(O)=O)(O)=O)O[C@H]1N(C=N2)C3=C2C(NCC4=CC=CC=C4)=NC=N3
CAS Number
1802226-78-3
Target & IC50
Others

Structure of PSB-12379, inhibitor

PSB-12379 Inhibitor – Cat# MBS5753736

Product References and Citations for PSB-12379, inhibitor

Bhattarai S, et al. alpha, beta-Methylene-ADP (AOPCP) Derivatives and Analogues: Development of Potent and Selective ecto-5'-Nucleotidase (CD73) Inhibitors. J Med Chem. 2015 Aug 13;58(15):6248-63.
Bhattarai S, et al. alpha, beta-Methylene-ADP (AOPCP) Derivatives and Analogues: Development of Potent and Selective ecto-5'-Nucleotidase (CD73) Inhibitors. J Med Chem. 2015 Aug 13;58(15):6248-63.

Other Notes

Small volumes of PSB-12379, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for PSB-12379 purchase

MBS5753736 is an inhibitor targeting PSB-12379.
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