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c(phg-isoDGR-(NMe)k) Inhibitor – C(phg-Isodgr-(Nme)k) TFA

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5754276

c(phg-isoDGR-(NMe)k) TFA is a potent and selective alpha5beta1-integrin ligand (IC50: 2.9nM). More details

Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
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Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
c(phg-isoDGR-(NMe)k) TFA, Inhibitor
Full Product Name
c(phg-isoDGR-(NMe)k) TFA
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
717.69
Solubility
DMSO: 250mg/mL (348.34mM) Need ultrasonic
(<1mg/ml refers to the product slightly soluble or insoluble)
Formula
C29H42F3N9O9
SMILES
O=C(CNC(C[C@@H](C(O)=O)NC([C@@H](C1=CC=CC=C1)NC([C@H]2CCCCN)=O)=O)=O)N[C@@H](CCCNC(N)=N)C(N2C)=O.OC(C(F)(F)F)=O
Target & IC50
alpha5beta1: ic50 2.9nM

Product References and Citations for c(phg-isoDGR-(NMe)k), inhibitor

Kapp TG, et al. N-Methylation of isoDGR Peptides: Discovery of a Selective alpha5beta1-Integrin Ligand as a Potent Tumor Imaging Agent. J Med Chem. 2018 Mar 22;61(6):2490-2499.
Kapp TG, et al. N-Methylation of isoDGR Peptides: Discovery of a Selective alpha5beta1-Integrin Ligand as a Potent Tumor Imaging Agent. J Med Chem. 2018 Mar 22;61(6):2490-2499.

Other Notes

Small volumes of c(phg-isoDGR-(NMe)k), inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for c(phg-isoDGR-(NMe)k) purchase

MBS5754276 is an inhibitor targeting c(phg-isoDGR-(NMe)k). Also known as c(phg-isoDGR-(NMe)k) TFA.
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