N6-Cyclopentyladenosine Inhibitor

Name: N6-Cyclopentyladenosine Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5755245
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5755245

N6-Cyclopentyladenosine (CPA) is a selective agonist of Adenosine A1 receptor (Ki: 2.3nM, 790nM and 43nM for human A1, A2A and A3 receptors, respectively). More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

N6-Cyclopentyladenosine, Inhibitor

Full Product Name

N6-Cyclopentyladenosine

Product Synonym Names

CPA; UK-80882

Form/Format

Solid. Powder

Purity/Purification

98.00%

Preparation and Storage

Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent

Molecular Weight

335.36

Solubility

DMSO: 12.5mg/mL (37.27mM) Need ultrasonic
(<1mg/ml refers to the product slightly soluble or insoluble)

Formula

C15H21N5O4

SMILES

OC[C@@H]1[C@H]([C@H]([C@H](N2C=NC3=C2N=CN=C3NC4CCCC4)O1)O)O

CAS Number

41552-82-3

Target & IC50

A1: ic50 2.3nM (ki)
A2A: ic50 790nM (ki)
A3: ic50 43nM (ki)

Product Categories/Family for N6-Cyclopentyladenosine, inhibitor

PI3K/Akt/mTOR signaling; mTOR; GPCR/G Protein

Product References and Citations for N6-Cyclopentyladenosine, inhibitor

Klotz KN, et al. Adenosine receptors and their ligands. Naunyn Schmiedebergs Arch Pharmacol. 2000 Nov;362(4-5):382-91.
Klotz KN, et al. Adenosine receptors and their ligands. Naunyn Schmiedebergs Arch Pharmacol. 2000 Nov;362(4-5):382-91.
Solino M, et al. Adenosine A1 receptor: A neuroprotective target in light induced retinal degeneration. PLoS One. 2018 Jun 18;13(6):e0198838.
Solino M, et al. Adenosine A1 receptor: A neuroprotective target in light induced retinal degeneration. PLoS One. 2018 Jun 18;13(6):e0198838.

Other Notes

Small volumes of N6-Cyclopentyladenosine, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for N6-Cyclopentyladenosine purchase

MBS5755245 is an inhibitor targeting N6-Cyclopentyladenosine.