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Indiplon Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5756719

Indiplon, a nonbenzodiazepine, hypnotic sedative, works by enhancing the action of the inhibitory neurotransmitter GABA, like most other nonbenzodiazepine sedatives. It primarily binds to the alpha1 subunits of the GABAA receptors in the brain. More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Product Name
Indiplon, Inhibitor
Full Product Name
Indiplon
Product Synonym Names
CL 285,489; CL-285,489; CL285,489; NBI 34060; NBI34060; NBI-34060; NBI-34060
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
376.43
Solubility
Water: Insoluble
DMSO: Soluble
(<1mg/ refers to the product slightly soluble or insoluble)
Formula
C20H16N4O2S
SMILES
CC(N(C)C1=CC=CC(C2=CC=NC3=C(C(C4=CC=CS4)=O)C=NN23)=C1)=O
CAS Number
325715-02-4

Product References and Citations for Indiplon, inhibitor

Shimizu M, Fukami T, Ito Y, Kurokawa T, Kariya M, Nakajima M, Yokoi T. Indiplon is hydrolyzed by arylacetamide deacetylase in human liver. Drug Metab Dispos. 2014 Apr;42(4):751-8. doi: 10.1124/dmd.113.056184. Epub 2014 Jan 24. PubMed PMID: 24464802.
Xu L, Wang J, Xiao B, Yang J, Liu Y, Huang R. Preparation and characterization of a novel polymorph of indiplon, Form alpha. Bioorg Med Chem Lett. 2012 Jan 15;22(2):963-8. doi: 10.1016/j. Bmcl.2011.12.013. Epub 2011 Dec 9. PubMed PMID: 22209207.
Lemon MD, Strain JD, Hegg AM, Farver DK. Indiplon in the management of insomnia. Drug Des Devel Ther. 2009 Sep 21;3:131-42. PubMed PMID: 19920929; PubMed Central PMCID: PMC2769245.
Marrs JC. Indiplon: a nonbenzodiazepine sedative-hypnotic for the treatment,of insomnia. Ann Pharmacother. 2008 Jul;42(7):1070-9. doi: 10.1345/aph.1K683. Epub 2008 Jul 1. PubMed PMID: 18594049.

Other Notes

Small volumes of Indiplon, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Indiplon purchase

MBS5756719 is an inhibitor targeting Indiplon.
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