Tropisetron Inhibitor

Name: Tropisetron Inhibitor; MyBioSource
Brand: MyBioSource
SKU: MBS5756952
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5756952

Tropisetron is a alpha7-nicotinic receptor agonist and 5-HT3 receptor antagonist with an IC50 of 70.1 +/- 0.9nM for 5-HT3 receptor. More details

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Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Tropisetron, Inhibitor

Full Product Name

Tropisetron

Product Synonym Names

ICS 205-930

Form/Format

Solid. Powder

Purity/Purification

98.00%

Preparation and Storage

Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent

Molecular Weight

284.35

Solubility

<1mg/ml refers to the product slightly soluble or insoluble

Formula

C17H20N2O2

SMILES

CN1C2CCC1CC(C2)OC(=O)C3=C[NH]C4=C3C=CC=C4

CAS Number

89565-68-4

Target & IC50

5-HT3 receptor: ic50 5.3nM (Ki)
alpha7 nAChR: ic50 6.9nM (Ki)

Product Categories/Family for Tropisetron, inhibitor

GPCR/G Protein; 5-HT Receptor; Neuroscience

Product References and Citations for Tropisetron, inhibitor

Macor JE, et al. Bioorg Med Chem Lett. 2001, 11(3):319-21.
Vega Lde L, et al. Biochem Pharmacol. 2005, 70(3):369-80.
Zirak MR, et al. Eur J Pharmacol. 2014, 738:222-9.

Other Notes

Small volumes of Tropisetron, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Tropisetron purchase

MBS5756952 is an inhibitor targeting Tropisetron.