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[Leu5]-Enkephalin TFA Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5758557

MBS5758557 is an inhibitor targeting [Leu5]-Enkephalin TFA. [Leu5]-Enkephalin is the most potent delta-receptor ago More details

Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
[Leu5]-Enkephalin TFA, Inhibitor
Full Product Name
[Leu5]-Enkephalin TFA
Product Synonym Names
Leu-enkephalin; Leucine enkephalin; Leucyl-enkephalin
Form/Format
Solid. Powder
Purity/Purification
98.00%
Preparation and Storage
Store at -20 degree C for 3 years powder
-80 degree C for 2 years in solvent
Molecular Weight
669.64
Solubility
<1mg/ml refers to the product slightly soluble or insoluble
Formula
C30H38F3N5O9
SMILES
CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)O.O=C(O)C(F)(F)F
CAS Number
73563-78-7
Target & IC50
delta-opioid receptor
Human Endogenous Metabolite

Product References and Citations for [Leu5]-Enkephalin TFA, inhibitor

Robert J Cassell, Krishna K Sharma, Hongyu Su,et al. The Meta-Position of Phe 4 in Leu-Enkephalin Regulates Potency, Selectivity, Functional Activity, and Signaling Bias at the Delta and Mu Opioid Receptors[J].Molecules, 24 (24) 2019 Dec 1
Robert J Cassell, Krishna K Sharma, Hongyu Su,et al. The Meta-Position of Phe 4 in Leu-Enkephalin Regulates Potency, Selectivity, Functional Activity, and Signaling Bias at the Delta and Mu Opioid Receptors[J].Molecules, 24 (24) 2019 Dec 1
Meunier J C, Moisand C. Binding of leu5-enkephalin and met5-enkephalin to a particulate fraction from rat cerebrum[J]. Febs Letters, 1977, 77(2):0-213.
Meunier J C, Moisand C. Binding of leu5-enkephalin and met5-enkephalin to a particulate fraction from rat cerebrum[J]. Febs Letters, 1977, 77(2):0-213.

Other Notes

Small volumes of [Leu5]-Enkephalin TFA, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.
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