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CPI-1205

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS848783

CPI-1205 is a highly potent (biochemical IC50 = 0.002 uM, cellular EC50 = 0.032 uM) and selective inhibitor of the histone lysine methyltransferase EZH2 (biochemical IC50 = 0.002 uM, cellular EC50 = 0.032 uM). Upon oral administration, CPI-1205 selectively… More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Product Name
CPI-1205, Biochemical
Full Product Name
CPI-1205
Product Synonym Names
N-[ (4-methoxy-6-methyl-2-oxo-1H-pyridin-3-yl) methyl]-2-methyl-1-[ (1R)-1-[1- (2; 2; 2-trifluoroethyl) piperidin-4-yl]ethyl]indole-3-carboxamide; CPI1205
Form/Format
Crystalline solid
Purity/Purification
>=98% by HPLC
Preparation and Storage
Store at -20 degree C
Shelf life: ~36 months
Molecular Weight
518.57
Solubility
>100 mg/ml in DMSO
Molecular Formula
C??H??F?N?O?
CAS Number
1621862-70-1
PubChem CID
78320408
SMILES
CC1=CC (=C (C (=O)N1)CNC (=O)C2=C (N (C3=CC=CC=C32)C (C)C4CCN (CC4)CC (F)(F)F)C)OC
InChi
InChI=1S/C27H33F3N4O3/c1-16-13-23 (37-4)21 (25 (35)32-16)14-31-26 (36)24-18 (3)34 (22-8-6-5-7-20 (22)24)17 (2)19-9-11-33 (12-10-19)15-27 (28,29)30/h5-8,13,17,19H,9-12,14-15H2,1-4H3, (H,31,36)(H,32,35)/t17-/m1/s1
InChi Key
HPODOLXTMDHLLC-QGZVFWFLSA-N

Product Categories/Family for CPI-1205 biochemical

Enzyme Inhibitors; Methyltransferase Inhibitors; Enzyme Inhibitors; Enzyme Inhibitors (A-Z); Biochemicals; Biochemicals (A-Z); Epigenetics; Epigenetic Modulators (A-Z); Epigenetics; Writer Enzymes; Protein Lysine Methyltransferases (PKMTs); PKMT Inhibitor

Structure of CPI-1205 biochemical

CPI-1205 Biochemical – Cat# MBS848783

Product References and Citations for CPI-1205 biochemical

https://pubchem.ncbi.nlm.nih.gov/compound/78320408

Other Notes

Small volumes of CPI-1205 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for CPI-1205 purchase

MBS848783 is a biochemical targeting CPI-1205.
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