Relacatib (SB-462795)

Name: Relacatib (SB-462795); MyBioSource
Brand: MyBioSource
SKU: MBS3604242
Price: 865 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3604242

Relacatib (SB-462795, GSK-462795) is a potent and orally bioavailable small molecule cathepsin inhibitor with Ki of 41, 68 and 53 pM for cathepsin K, L and V, respectively. More details

$865 / 5 mg +1 FREE 8GB USB

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Relacatib, Biochemical

Full Product Name

Relacatib

Product Synonym Names

SB-462795; GSK-462795

Purity/Purification

>98% (HPLC)

Preparation and Storage

Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack

Molecular Weight

540.635

Target

Cathepsin

Receptor

Cathepsin

Chemical Name

N-((S)-4-methyl-1-(((4S, 7R)-7-methyl-3-oxo-1-(pyridin-2-ylsulfonyl)azepan-4-yl)amino)-1-oxopentan-2-yl)benzofuran-2-carboxamide

SMILES

O=C(C1=CC2=CC=CC=C2O1)N[C@@H](CC(C)C)C(N[C@@H]3C(CN(S(=O)(C4=NC=CC=C4)=O)[C@H](C)CC3)=O)=O

Molecular Formula

C27H32N4O6S

CAS Number

362505-84-8

Product Categories/Family for Relacatib biochemical

Osteoporosis; Metabolic Enzyme/Protease; Metabolic Disease

Product References and Citations for Relacatib biochemical

1. Yamashita DS, et al. J Med Chem. 2006 Mar 9; 49 (5):1597-612.
2. Kumar S, et al. Bone. 2007 Jan; 40 (1):122-31.

Other Notes

Small volumes of Relacatib biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Relacatib purchase

MBS3604242 is a biochemical targeting Relacatib.