Relugolix (TAK385)

Name: Relugolix (TAK385); MyBioSource
Brand: MyBioSource
SKU: MBS3607580
Price: 220 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3607580

Relugolix is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, with potential antineoplastic activity. More details

$220 / 2 mg +1 FREE 8GB USB

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

Relugolix, Biochemical

Full Product Name

Relugolix

Product Synonym Names

TAK385; TAK-385; TAK 385; Relugolix

Purity/Purification

>98% (HPLC)

Preparation and Storage

Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack

Molecular Weight

623.63

Suitability

DMSO: 50mg/mL (80.18mM)

Target

MDM2-p53

Receptor

GNRHR

Chemical Name

1-(4-(1-(2, 6-difluorobenzyl)-5-((dimethylamino)methyl)-3-(6-methoxypyridazin-3-yl)-2, 4-dioxo-1, 2, 3, 4-tetrahydrothieno[2, 3-d]pyrimidin-6-yl)phenyl)-3-methoxyurea

SMILES

CN(C)Cc1c(sc2c1c(=O)n(c(=O)n2Cc1c(cccc1F)F)c1nnc(cc1)OC)c1ccc(cc1)NC(=O)NOC

Molecular Formula

C29H27F2N7O5S

CAS Number

737789-87-6

Product Categories/Family for Relugolix biochemical

Apoptosis; Cancer

Product References and Citations for Relugolix biochemical

1. MacLean DB et al. J Clin Endocrinol Metab. 2015 Dec; 100 (12):4579-87.

Other Notes

Small volumes of Relugolix biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for Relugolix purchase

MBS3607580 is a biochemical targeting Relugolix.