BRD32048 Inhibitor

BRD32048 is a top candidate ETV1 perturbagen. BRD32048 inhibits p300-dependent acetylation of ETV1, thereby promoting its degradation.

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1 Kollaredd M Sherrar A Par JH Szeme M Gallache K Meleg Z Oltea S Michaeli M Cinat Jr Kaid A Mali K Th smal molecul inhibito YK-4-27 disrupt mitoti progressio o neuroblastom cells overcome dru resistanc an synergize wit inhibitor o mitosis Cance Lett 201 Se 10 03:74-85 doi 10.1016/j.canlet.2017.05.027 Epu 201 Ju 7 PubMe PMID 28602975 PubMe Centra PMCID PMC5542135 href="javascript:void(0) rel="nofollow >
2 Po MS Stransk N Garvi CW Theurilla JP Hartma EC Lewi TA Zhon C Culyb EK Li F Daniel DS Pagliarin R Ronc L Koehle AN Garrawa LA smal molecul tha bind an inhibit th ETV transcriptio facto oncoprotein Mo Cance Ther 201 Jun 3(6):1492-502 doi 10.1158/1535-7163.MCT-13-0689 Epu 201 Ap 15 PubMe PMID 24737027 PubMe Centra PMCID PMC4154495.

Small volumes of BRD32048, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

MBS5773585 is an inhibitor targeting BRD32048.