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BRD7-IN-1 Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5770567

BRD7-IN-1, a modified derivative of BI7273 (BRD7/9 inhibitor), binds to a VHL ligand via a linker to form a PROTAC VZ185 (VZ185 against BRD7/9 with DC50s of 4.5 and 1.8nM, respectively). More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
BRD7-IN-1, Inhibitor
Full Product Name
BRD7-IN-1
Product Gene Name
BRD7-IN-1, inhibitor
Purity/Purification
98%
Preparation and Storage
Powder: -2 degree C for 3 years
In solvent: -80 degree C for 2 years
Molecular Weight
467.39
SMILES
CN1C=C(C2=CC(OC)=C(CN3CCNCC3)C(OC)=C2)C(C=CN=C4)=C4C1=O.Cl.Cl
Formula
C22H28Cl2N4O3
Target
Epigenetic Reader Domain
Solubility
DMSO: 30mg/mL (64.19 mM),
Need ultrasonic
H2O: 100mg/mL (213.95 mM),
Need ultrasonic
(<1mg/mL refers to the product slightly soluble or insoluble)

Product Categories/Family for BRD7-IN-1, inhibitor

Chromatin/Epigenetic

Structure of BRD7-IN-1, inhibitor

BRD7-IN-1, CAS MBS5770567
BRD7-IN-1 Inhibitor – Cat# MBS5770567

Structure of BRD7-IN-1, inhibitor

BRD7-IN-1, CAS MBS5770567
BRD7-IN-1 Inhibitor, Structure – Cat# MBS5770567

Product References and Citations for BRD7-IN-1, inhibitor

1 Zopp V e al Iterativ Desig an Optimizatio o Initiall Inactiv Proteolysi Targetin Chimera (PROTACs Identif VZ18 a Potent Fast an Selectiv vo Hippel-Linda (VHL Base Dua Degrade Prob o BRD an BRD7 Me Chem 201 Ja 24 2(2):699-726.

Other Notes

Small volumes of BRD7-IN-1, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for BRD7-IN-1 purchase

MBS5770567 is an inhibitor targeting BRD7-IN-1.
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