Dafphedyn Inhibitor

Dafphedyn, [D-Ala2, (F5) Phe4]-dynorphin 1-13-NH2 (DAFPHEDYN) is an effective analog of strong endorphin 1-13 and produces diuretic and deep analgesia when administered intravenously in rats.

1 Walke JM Co DH Youn EA Baldrigh G Siege SF Bowe WD Aki H [D-Ala2 (F5 Phe]-dynorphi 1-13-NH (DAFPHEDYN) poten analo o dynorphi 1-13 Peptides 198 Sep-Oct (5):811-7 PubMe PMID 2893357.
2 Gosnel BA Majchrza MJ Krah DD Effect o preferentia delt an kapp opioi recepto agonist o th intak o hypotoni saline Physio Behav 199 Mar 7(3):601-3 PubMe PMID 1972796.
3 Kostrzew RM Bru R Co DH Criswel H Cooga PS Kasti AJ D-Ala2,F5Phe4-dynorphi amide a opiat wit analgesi an toxi properties Po Pharmaco Pharm 199 Mar-Apr 4(2):109-20 PubMe PMID 1357636.
4 Soli AV Lyashe AY Lyashe YD Effect o Opioi Peptide o Change i Lipi Metabolis i Rat Subjecte t Swimmin Stress Bul Ex Bio Med 201 Jan 62(3):313-315 doi 10.1007/s10517-017-3603-7 Epu 201 Ja 14 PubMe PMID 28091903.

Small volumes of Dafphedyn, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

MBS5780810 is an inhibitor targeting Dafphedyn.