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GV-196771A Inhibitor

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS5766776

MBS5766776 is an inhibitor targeting GV-196771A. GV-196771A, a sodium salt form of GV196771, is annMDA receptor antagonist. More details

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Product Documentation
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Sample Manual Insert View PDF
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Testing Data View PDF
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Certificate of Analysis (COA) View PDF
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QC Report View PDF
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Material Safety Data Sheet View PDF
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Technical Datasheet View PDF
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Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
GV-196771A, Inhibitor
Full Product Name
GV-196771A
Product Gene Name
GV-196771A, inhibitor
Purity/Purification
98%
Preparation and Storage
Powder: -2 degree C for 3 years
In solvent: -80 degree C for 2 years
Molecular Weight
423.22
SMILES
[Na+].[O-]C(=O)c1[nH]c2cc(Cl)cc(Cl)c2c1\C=C1/CCN(C1=O)c1ccccc1
Formula
C20H13Cl2N2NaO3
CAS Number
166974-23-8
Target
Others
Solubility
(<1mg/mL refers to the product slightly soluble or insoluble)
In_vitro
GV196771 is annMDA receptor antagonist with low oral bioavailability in rats and mice. GV196771 has low oral bioavailability (<10%) and plasma clearance (~2 mL/min/kg) in rats. GV196771 is a potent antagonist of the modulatory glycine site of the N-methyl-D-aspartate receptor. GV196771 is a potent antagonist of the modulatory glycine site of thenMDA receptor developed for treatment of neuropathic pain.

Product Categories/Family for GV-196771A, inhibitor

Others

Structure of GV-196771A, inhibitor

GV-196771A, CAS 166974-23-8
GV-196771A Inhibitor – Cat# MBS5766776

Structure of GV-196771A, inhibitor

GV-196771A, CAS 166974-23-8
GV-196771A Inhibitor, Structure – Cat# MBS5766776

Product References and Citations for GV-196771A, inhibitor

1 Poll JW e al Th systemi exposur o a N-methyl-D-aspartat recepto antagonis i limite i mic b th P-glycoprotei an breas cance resistanc protei efflu transporters Dru Meta Dispos 200 Jul 2(7):722-6.

Other Notes

Small volumes of GV-196771A, inhibitor vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.
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