Chemical structure of KT5720 (SIH-457), a PKA kinase inhibitor. CAS #: 108068-98-0. Molecular Formula: C32H31N3O5. Molecular Weight: 537.6 g/mol.

KT5720 Small Molecule

Name: KT5720 Small Molecule; MyBioSource
Brand: MyBioSource
SKU: MBS808157
Price: 310 USD
Availability: InStock
Rating: 5 (10 reviews)

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS808157

KT5720 is a potent and selective inhibitor of protein kinase A (PKA). This compound blocks PKA signaling through competitive inhibition. It causes no significant effect on protein kinase C (PKC), protein kinase G (PKG) or myosin light chain kinase (mlCK).… More details

$310 / 0.1 mg +1 FREE 8GB USB

Product Documentation

Sample Manual Insert View PDF

Testing Data View PDF

Certificate of Analysis (COA) View PDF

QC Report View PDF

Material Safety Data Sheet View PDF

Technical Datasheet View PDF

Protocol View PDF

Product Overview

Online Datasheet in PDF

Product Name

KT5720, Small Molecule

Full Product Name

KT5720

Product Gene Name

KT5720 small molecule

Product Synonym Names

PKA kinase inhibitor; (9S,10S,12R)-2,3,9,10,11,12-Hexahydro-10-hydroxy-9-methyl-1-oxo-9,12-epoxy-1H-diindolo[1,2,3-fg:3',2',1'-kl]pyrrolo[3,4-i][1,6]benzodiazocine-10-carboxylic acid hexyl ester

Host

Synthetic

Form/Format

White powder

Purity/Purification

>=98% (TLC)

Preparation and Storage

Store at -20 degree C.

Molecular Weight

537.6

Solubility

Soluble in methanol: clear colorless solution at 5 mg/ml

CAS Number

108068-98-0

Molecular Formula

C32H31N3O5

SMILES

[N]47C1=C(C6=C(C2=C1[N](C3=CC=CC=C23)[C@H]5O[C@@]4([C@](C5)(O)C(=O)OCCCCCC)C)C(NC6)=O)C8=C7C=CC=C8

InChI

1S/C32H31N3O5/c1-3-4-5-10-15-39-30(37)32(38)16-23-34-21-13-8-6-11-18(21)25-26-20(17-33-29(26)36)24-19-12-7-9-14-22(19)35(28(24)27(25)34)31(32,2)40-23/h6-9,11-14,23,38H,3-5,10,15-17H2,1-2H3,(H,33,36)

InChI Key

ZHEHVZXPFVXKEY-UHFFFAOYSA-N

PubChem CID

3844

Product Categories/Family for KT5720 small molecule

Small Molecules; Inhibitor; Cell Signaling; Cancer; Apoptosis; Cancer Growth Inhibitors; Tyrosine Kinase Inhibitors

Product References and Citations for KT5720 small molecule

1. Kase H., et al. (1987) Biochem. Biophys. Res. Comm. 142(2): 436-440. 2. Gadbois D.M., Crissman H.A., Tobey R.A., & Bradbury E.M. (1992) Pro. Na. Aca. Sci. USA. 89(18): 8626-8630.

Other Notes

Small volumes of KT5720 small molecule vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for KT5720 purchase

MBS808157 is a small molecule targeting KT5720. Host: Synthetic.