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GSK-256066

For Research Use Only. Not for use in diagnostic procedures. Catalog #: MBS3605998

A potent, selective PDE4 inhibitor with pIC50 of 11.5, 11.3, 11.4, and 11.9 for PDE4B, A, C, and D, respectively. More details

$235 / 2 mg +1 FREE 8GB USB
Product Documentation
PDF
Sample Manual Insert View PDF
PDF
Testing Data View PDF
PDF
Certificate of Analysis (COA) View PDF
PDF
QC Report View PDF
PDF
Material Safety Data Sheet View PDF
PDF
Technical Datasheet View PDF
PDF
Protocol View PDF

Product Overview

Online Datasheet in PDF
Product Name
GSK-256066, Biochemical
Full Product Name
GSK-256066
Product Synonym Names
GSK256066; GSK 256066
Purity/Purification
>98% (HPLC)
Preparation and Storage
Store at -20 degree C
Stability: >=2 years
Shipping: Ice Pack
Molecular Weight
518.5842
Suitability
DMSO: >=5.2mg/mL
Target
PDE
Receptor
PDE4B
Chemical Name
3-Quinolinecarboxamide, 6-[[3-[(dimethylamino)carbonyl]phenyl]sulfonyl]-4-[(3-methoxyphenyl)amino]-8-methyl
SMILES
CC1=CC(=CC2=C(C(=CN=C12)C(=O)N)NC3=CC(=CC=C3)OC)S(=O)(=O)C4=CC=CC(=C4)C(=O)N(C)C
Molecular Formula
C27H26N4O5S
CAS Number
801312-28-7

Product Categories/Family for GSK-256066 biochemical

COPD; Angiogenesis; Inflammation/Immunology

Structure of GSK-256066 biochemical

GSK-256066 Biochemical – Cat# MBS3605998

Product References and Citations for GSK-256066 biochemical

1. Woodrow MD, et al. Bioorg Med Chem Lett. 2009 Sep 1; 19 (17):5261-5.
2. Tralau-Stewart CJ, et al. J Pharmacol Exp Ther. 2011 Apr; 337 (1):145-54.
3. Nials AT, et al. J Pharmacol Exp Ther. 2011 Apr; 337 (1):137-44.

Other Notes

Small volumes of GSK-256066 biochemical vial(s) may occasionally become entrapped in the seal of the product vial during shipment and storage. If necessary, briefly centrifuge the vial on a tabletop centrifuge to dislodge any liquid in the container`s cap. Certain products may require to ship with dry ice and additional dry ice fee may apply.

Searchable Terms for GSK-256066 purchase

MBS3605998 is a biochemical targeting GSK-256066.
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